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Ivankin, DI, Kornienko, TE, Mikhailova, MA, Dyrkheeva, NS, Zakharenko, AL, Achara, C, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Golyshev, VM, Luzina, OA, Volcho, KP, Salakhutdinov, NF and Lavrik, OI
(2023)
Novel TDP1 Inhibitors: Disubstituted Thiazolidine-2,4-Diones Containing Monoterpene Moieties.
International Journal of Molecular Sciences, 24 (4).
Ivankin, DI, Dyrkheeva, NS, Zakharenko, AL, Ilina, ES, Zarkov, TO, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Luzina, OA, Volcho, KP, Salakhutdinov, NF and Lavrik, OI
(2022)
Monoterpene substituted thiazolidin-4-ones as novel TDP1 inhibitors: Synthesis, biological evaluation and docking.
Bioorganic & Medicinal Chemistry Letters, 73 (128909).
Munkuev, AA, Dyrkheeva, NS, Kornienko, TE, Ilina, ES, Ivankin, DI, Suslov, EV, Korchagina, DV, Gatilov, YV, Zakharenko, AL, Malakhova, AA, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Volcho, KP, Salakhutdinov, NF and Lavrik, OI
(2022)
Adamantane-Monoterpenoid Conjugates Linked via Heterocyclic Linkers Enhance the Cytotoxic Effect of Topotecan.
Molecules, 27 (11).
Salomatina, OV, Dyrkheeva, NS, Popadyuk, II, Zakharenko, AL, Ilina, ES, Komarova, NI, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Salakhutdinov, NF, Lavrik, OI and Volcho, KP
(2021)
New Deoxycholic Acid Derived Tyrosyl-DNA Phosphodiesterase 1 Inhibitors Also Inhibit Tyrosyl-DNA Phosphodiesterase 2.
Molecules, 27 (1).
Dyrkheeva, NS, Filimonov, AS, Luzina, OA, Zakharenko, AL, Ilina, ES, Malakhova, AA, Medvedev, SP, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Volcho, KP, Zakian, SM, Salakhutdinov, NF and Lavrik, OI
(2021)
New Hybrid Compounds Combining Fragments of Usnic Acid and Monoterpenoids for Effective Tyrosyl-DNA Phosphodiesterase 1 Inhibition.
Biomolecules, 11 (7).
Munkuev, AA, Mozhaitsev, ES, Chepanova, AA, Suslov, EV, Korchagina, DV, Zakharova, OD, Ilina, ES, Dyrkheeva, NS, Zakharenko, AL, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Volcho, KP, Salakhutdinov, NF and Lavrik, OI
(2021)
Novel Tdp1 Inhibitors Based on Adamantane Connected with Monoterpene Moieties via Heterocyclic Fragments.
Molecules, 26 (11).
pp. 1-23.
Gladkova, ED, Nechepurenko, IV, Bredikhin, RA, Chepanova, AA, Zakharenko, AL, Luzina, OA, Ilina, ES, Dyrkheeva, NS, Mamontova, EM, Anarbaev, RO, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Volcho, KP, Salakhutdinov, NF and Lavrik, OI
(2020)
The First Berberine-Based Inhibitors of Tyrosyl-DNA Phosphodiesterase 1 (Tdp1), an Important DNA Repair Enzyme.
International Journal of Molecular Sciences, 21 (19).
Il'ina, IV, Dyrkheeva, NS, Zakharenko, AL, Sidorenko, AY, Li-Zhulanov, NS, Korchagina, DV, Chand, R, Ayine-Tora, DM, Chepanova, AA, Zakharova, OD, Ilina, ES, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Malakhova, AA, Medvedev, SP, Zakian, SM, Volcho, KP, Salakhutdinov, NF and Lavrik, OI
(2020)
Design, Synthesis, and Biological Investigation of Novel Classes of 3-Carene-Derived Potent Inhibitors of TDP1.
Molecules, 25 (15).
Mamontova, EM, Zakharenko, AL, Zakharova, OD, Dyrkheeva, NS, Volcho, KP, Reynisson, J
ORCID: https://orcid.org/0000-0003-4174-9512, Arabshahi, HJ, Salakhutdinov, NF and Lavrik, OI
(2019)
Identification of novel inhibitors for the tyrosyl-DNA-phosphodiesterase 1 (Tdp1) mutant SCAN1 using virtual screening.
Bioorganic & Medicinal Chemistry, 28 (1).
115234 - ?.
Filimonov, AS, Chepanova, AA, Luzina, OA, Zakharenko, AL, Zakharova, OD, Ilina, ES, Dyrkheeva, NS, Kuprushkin, MS, Kolotaev, AV, Khachatryan, DS, Patel, J, Leung, IKH, Chand, R, Ayine-Tora, DM, Reynisson, J, Volcho, KP, Salakhutdinov, NF and Lavrik, OI (2019) New Hydrazinothiazole Derivatives of Usnic Acid as Potent Tdp1 Inhibitors. Molecules, 24 (20).

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